Sulfamethoxazole

Category: pharmacological

Aliases: Component of Bactrim / Septra

Pharmacological Mechanism

Sulfonamide antibiotic — competitive inhibitor of bacterial dihydropteroate synthase (DHPS) blocking folate synthesis. Always co-formulated with trimethoprim for synergistic folate-pathway blockade. CYP2C9 inhibitor (raises warfarin INR).

Half-Life (t½)

PO: 10h, IV: 10h

Dosing Guidelines

Target Organ Systems