Remifentanil

Category: pharmacological

Aliases: Ultiva

Pharmacological Mechanism

Ultra-short-acting synthetic μ-opioid agonist — esterase-cleared (not CYP) giving ~3-4 min context-sensitive half-time even after long infusions. IV-only continuous infusion for surgical anesthesia. Rapid offset means no opioid-tolerance build-up across surgery.

Half-Life (t½)

IV: 0.16h

Dosing Guidelines

Target Organ Systems