Rapamycin
Category: other
Aliases: sirolimus
Pharmacological Mechanism
mTORC1 inhibitor (FKBP12 complex); chronic mTORC2 inhibition with sustained dosing.
Half-Life (t½)
PO: 62h
Dosing Guidelines
- PO: Typical 6mg (Range: 1 - 8 )
Target Organ Systems
- immune-hematologic
- musculoskeletal