Methandrostenolone

Category: hormone

Aliases: Dianabol, Dbol, methandienone, metandienone

Pharmacological Mechanism

17α-methylated Δ1-testosterone analog; an orally active AR agonist (the 17α-methyl resists hepatic first-pass, enabling PO use but conferring hepatotoxicity). Strongly anabolic with moderate androgenicity; aromatizes to 17α-methylestradiol (estrogenic — gynecomastia, water retention). Classic oral "kickstart" with 17αα-related liver strain and HPG suppression.

Dosing Guidelines

Target Organ Systems

Notes

PubChem CID 6300. No primary abstract names a methandienone plasma half-life (the "3–6 h" figure traces only to secondary pages); no verbatim AR Ki (see AUTHORING_GAPS). digestive = hepatic 17αα strain.

Chemical Identifiers