Mesterolone

Category: hormone

Aliases: Proviron

Pharmacological Mechanism

Orally active 1α-methyl dihydrotestosterone derivative; not 17α-alkylated (low hepatotoxicity). Weak anabolic; used as an androgen/anti-estrogen adjunct that binds SHBG and the androgen receptor, raising free testosterone and adding androgenic "hardening" without aromatization.

Dosing Guidelines

Target Organ Systems