Luteolin

Category: flavonoid

Aliases: 3',4',5,7-Tetrahydroxyflavone

Pharmacological Mechanism

Flavone with strong mast-cell-stabilising activity and microglial anti-inflammation (blocks IFN-γ-induced microglial activation). PDE4 inhibition contributes to anti-inflammatory profile. Attenuates oxidative stress via Nrf2 pathway.

Half-Life (t½)

PO: 3h

Dosing Guidelines

Target Organ Systems