Larazotide

Category: peptide

Aliases: AT-1001

Pharmacological Mechanism

Zonulin antagonist octapeptide — blocks zonulin-induced tight-junction disassembly in gut epithelium. Trialed for celiac disease as adjunct to gluten-free diet (failed Phase 3 in 2022); biohacker / leaky-gut interest persists.

Half-Life (t½)

PO: 1h

Dosing Guidelines

Target Organ Systems