Kojic Acid

Category: topical

Aliases: 5-Hydroxy-2-(hydroxymethyl)-4H-pyran-4-one

Pharmacological Mechanism

Fungal metabolite (Aspergillus oryzae — koji rice fermentation). Chelates copper at tyrosinase active site → inhibits melanin synthesis. Less effective but less irritating than hydroquinone; paired with azelaic acid / glycolic acid in fading stacks.

Target Organ Systems