Cisplatin

Category: pharmacological

Pharmacological Mechanism

Platinum-based DNA crosslinker — covalently binds N7 of guanine forming intra- and inter-strand adducts that block DNA replication. Backbone of testicular, lung, head-and-neck, ovarian regimens. Nephrotoxicity, ototoxicity, severe nausea — pre-medication with antiemetics + IV hydration mandatory.

Half-Life (t½)

IV: 80h

Dosing Guidelines

Target Organ Systems