Ceftriaxone

Category: pharmacological

Aliases: Rocephin

Pharmacological Mechanism

Third-generation cephalosporin β-lactam — extended gram-negative + good gram-positive coverage. Once-daily IV/IM dosing makes it a workhorse for inpatient pneumonia, meningitis (CSF penetration), gonorrhea single-dose. Biliary > renal clearance — sludging in gallbladder.

Half-Life (t½)

IV: 8h, IM: 8.1h

Dosing Guidelines

Target Organ Systems