Capsaicin

Category: alkaloid

Aliases: Capsicum, Chili extract

Pharmacological Mechanism

TRPV1 agonist — initial activation produces burning sensation; chronic exposure desensitizes nociceptors → topical analgesia for neuropathic pain (post-herpetic, diabetic neuropathy). Oral capsicum used for thermogenic / metabolic supplementation; modest effect.

Half-Life (t½)

TD: 24h

Dosing Guidelines

Target Organ Systems